Tocris™ A 366

Potent and selective G9a/GLP inhibitor

Manufacturer: Tocris™ 5163/50

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Catalog No. 51-635-0

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For Research Use Only


    Product Type A 366
    Inhibitors A 366
    Purity >98
    Molecular Weight 329.44
    Quantity 50mg

    Potent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50 = 3.3nM). Exhibits >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. Decreases levels of lysine 9 dimethylation on histone H3 (H3K9Me2) in PC3 cells.

    • Chemical Name: 5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine
    • Formula: C19H27N3O2
    • CAS Number: 1527503-11-2
    • Solubility: Soluble to 100mM in 1eq. HCl and to 100mM in DMSO
    • Purity: >98

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