Tocris A 366
Potent and selective G9a/GLP inhibitor
Manufacturer: Tocris 5163/10
DescriptionPotent and selective G9a/GLP histone lysine methyltransferase inhibitor (IC50 = 3.3nM). Exhibits >1000-fold selectivity for G9a/GLP over 21 other methyltransferases. Decreases levels of lysine 9 dimethylation on histone H3 (H3K9Me2) in PC3 cells.
- Chemical Name: 5'-Methoxy-6'-[3-(1-pyrrolidinyl)propoxy]spiro[cyclobutane-1,3'-[3H]indol]-2'-amine
- Formula: C19H27N3O2
- CAS Number: 1527503-11-2
- Solubility: Soluble to 100mM in 1eq. HCl and to 100mM in DMSO
- Purity: >98
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