Uncompetitive Epac1 inhibitor
Manufacturer: Tocris 4793/10
DescriptionUncompetitive Epac1 inhibitor. Blocks Epac-induced Rap activation and prevents isoprenaline-induced autophagy flux in cardiomyocytes. Has no effect on PKA activity in the presence of cAMP.
- Chemical Name: 5,7-Dibromo-6-fluoro-3,4-dihydro-2-methyl-1(2H)-quinolinecarboxaldehyde
- Formula: C11H10Br2FNO
- CAS Number: 143703-25-7
- Solubility: Soluble to 100mM in DMSO and to 50mM in ethanol
- Purity: >98