Tocris Bioscience CID 16020046
Selective GPR55 antagonist
Manufacturer: Tocris Bioscience 4959/10
DescriptionSelective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21µM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase,µ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.
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For Research Use Only