CID 16020046, Tocris Bioscience
Selective GPR55 antagonist
Manufacturer: Tocris Bioscience 4959/25
DescriptionSelective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21 μM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase, μ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.
|Observed MW: 425.44|
Safety and Handling
Recommended Storage : Store at 4°C
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