Tocris™ CID 16020046

Selective GPR55 antagonist

Manufacturer: Tocris™ 4959/10

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Catalog No. 49-591-0R

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For Research Use Only


    Specifications

    Product Type CID 16020046
    Inhibitors CID 16020046
    Purity >99
    Molecular Weight 425.44
    Quantity 10mg

    Selective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21µM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase,µ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.

    • Chemical Name: 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
    • Formula: C25H19N3O4
    • CAS Number: 834903-43-4
    • Solubility: Soluble to 100mM in DMSO
    • Purity: >99

  • Description & Specifications

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