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Tocris™ CID 16020046

Selective GPR55 antagonist

Manufacturer:  Tocris™ 4959/10

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Catalog No. 49-591-0R


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For Research Use Only


Specifications

Description

Selective GPR55 antagonist. Inhibits LPI-induced Ca2+ signaling (IC50 = 0.21µM in HEK-GPR55 cells), ERK1/2 phosphorylation and GPR55-mediated transcription factor activation. Displays weak inhibition of acetylcholinesterase,µ-opioid receptor, KCNH2 and hERG. Decreases LPI-induced GPR55 internalization. Reduces experimental intestinal inflammation in mice.
  • Chemical Name: 4-[4,6-Dihydro-4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxopyrrolo[3,4-c]pyrazol-5(1H)-yl]benzoic acid
  • Formula: C25H19N3O4
  • CAS Number: 834903-43-4
  • Solubility: Soluble to 100mM in DMSO
  • Purity: >99
Description & Specifications

Specifications

CID 16020046
>99
10mg
CID 16020046
425.44
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