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GP 1a, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
511532-96-0
C23H22Cl2N4O
441.356
FNOMTMVRTBHRET-UHFFFAOYSA-N
gp 1a,n-piperidin-1-yl-1-2,4-dichlorophenyl-1,4-dihydro-6-methylindeno 1,2-c pyrazole-3-carboxamide,6-methyl-1-2,4-dichlorophenyl-n-piperidin-1-yl-1,4-dihydroindeno 1,2-c pyrazole-3-carboxamide
10252734
1-(2,4-dichlorophenyl)-6-methyl-N-piperidin-1-yl-4H-indeno[1,2-c]pyrazole-3-carboxamide
CC1=CC2=C(C=C1)C3=C(C2)C(=NN3C4=C(C=C(C=C4)Cl)Cl)C(=O)NN5CCCCC5
This item is not returnable. View return policy
511532-96-0
C23H22Cl2N4O
441.356
FNOMTMVRTBHRET-UHFFFAOYSA-N
gp 1a,n-piperidin-1-yl-1-2,4-dichlorophenyl-1,4-dihydro-6-methylindeno 1,2-c pyrazole-3-carboxamide,6-methyl-1-2,4-dichlorophenyl-n-piperidin-1-yl-1,4-dihydroindeno 1,2-c pyrazole-3-carboxamide
10252734
1-(2,4-dichlorophenyl)-6-methyl-N-piperidin-1-yl-4H-indeno[1,2-c]pyrazole-3-carboxamide
CC1=CC2=C(C=C1)C3=C(C2)C(=NN3C4=C(C=C(C=C4)Cl)Cl)C(=O)NN5CCCCC5

Highly selective CB2 agonist

CB 2 receptor inverse agonist (pEC 50 = 7.1), shown in cAMP, GTPγS and β-arrestin recruitment assays. Demonstrates approximately 30-fold selectivity for CB 2 receptors over CB 1 receptors. Increases P-ERK1/2 expression in HL-60 cells in vitro.
Quantity 50mg
Assay Percent Range >99%
Formula Weight 441.35
Chemical Name or Material GP 1a

Recommended Storage : Store at Room Temperature