Tocris GSK 5959
Potent and selective BRPF1 inhibitor
Manufacturer: Tocris 5385/50
DescriptionPotent and selective BRPF1 bromodomain inhibitor (IC50 = 80nM). Exhibits >100-fold selectivity for BRPF1 over a panel of 35 other bromodomains, including BRPF2/3 and BET family bromodomains. Inhibits BRPF1 interaction with histone H3.3. Cell permeable.
- Chemical Name: N-[2,3-Dihydro-1,3-dimethyl-2-oxo-6-(1-piperidinyl)-1H-benzimidazol-5-yl]-2-methoxybenzamide
- Formula: C22H26N4O3
- CAS Number: 901245-65-6
- Solubility: Soluble to 10mM in DMSO with sonication
- Purity: >99
We continue to work to improve your shopping experience and your feedback regarding this content is very important to us. Please use the form below to provide feedback related to the content on this product.
Your feedback has been submitted. Fisher Scientific is always working to improve our content for you. We appreciate your feedback.Ok