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JNJ 16259685, Tocris Bioscience™
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Quantity:
10 mg
50 mg
Description
Sub-nanomolar potent, non-competitive mGlu1 antagonist (Ki = 0.34 nM). Inhibits glutamate-induced Ca2+ response at the human mGlu1 receptor with an IC50 value of 0.55 nM. Selective over mGlu5 (> 400-fold) and displays no activity at mGlu2, mGlu3, mGlu4, mGlu6, AMPA or NMDA receptors (IC50 > 10 μM). Centrally active following systemic administration.
Specifications
Quantity | 10 mg |
Formula Weight | 325.41 |
Percent Purity | >98% |
Chemical Name or Material | JNJ 16259685 |
Safety and Handling
Recommended Storage | Store at +4°C |
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