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Tocris™ OF 1

Selective BRPF1B and BRPF2 inhibitor

Manufacturer:  Tocris™ 5289/50

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Catalog No. 52-895-0

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For Research Use Only



Selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500nM respectively). Exhibits 39-fold selectivity for BRPF1B and BRPF2 over BRD4. Accelerates FRAP recovery at 5µM in a BRPF2 FRAP assay.
  • Chemical Name: 4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide
  • Formula: C17H18BrN3O4S
  • CAS Number: 919973-83-4
  • Solubility: Soluble to 20mM in DMSO
  • Purity: >98
Description & Specifications


OF 1
OF 1
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