Tocris™ OF 1

Selective BRPF1B and BRPF2 inhibitor

Manufacturer: Tocris™ 5289/10

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Catalog No. 52-891-0

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    Inhibitors OF 1
    Purity >98
    Molecular Weight 440.31
    Quantity 10mg
    Product Type OF 1

    Selective BRPF1B and BRPF2 bromodomain inhibitor (Kd values are 100 and 500nM respectively). Exhibits 39-fold selectivity for BRPF1B and BRPF2 over BRD4. Accelerates FRAP recovery at 5µM in a BRPF2 FRAP assay.

    • Chemical Name: 4-Bromo-N-(2,3-dihydro-6-methoxy-1,3-dimethyl-2-oxo-1H-benzimidazol-5-yl)-2-methylbenzenesulfonamide
    • Formula: C17H18BrN3O4S
    • CAS Number: 919973-83-4
    • Solubility: Soluble to 20mM in DMSO
    • Purity: >98

  • Description & Specifications

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