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PD 135158, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
130285-87-9
C35H44N4O6
616.759
NNTPEWZUKRSTMM-VVUNRPKCSA-N
4-r-2-r-2-1s,4beta-1,7,7-trimethylbicyclo 2.2.1 heptan-2alpha-yl oxycarbonylamino-2-methyl-3-1h-indol-3-yl propanoylamino-1-phenylethylamino-4-oxobutyric acid
92211238
4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-2-[[(1S,3R,4S)-4,7,7-trimethyl-3-bicyclo[2.2.1]heptanyl]oxycarbonylamino]propanoyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid
CC1(C2CCC1(C(C2)OC(=O)NC(C)(CC3=CNC4=CC=CC=C43)C(=O)NCC(C5=CC=CC=C5)NC(=O)CCC(=O)O)C)C
This item is not returnable. View return policy
130285-87-9
C35H44N4O6
616.759
NNTPEWZUKRSTMM-VVUNRPKCSA-N
4-r-2-r-2-1s,4beta-1,7,7-trimethylbicyclo 2.2.1 heptan-2alpha-yl oxycarbonylamino-2-methyl-3-1h-indol-3-yl propanoylamino-1-phenylethylamino-4-oxobutyric acid
92211238
4-[[(1R)-2-[[(2R)-3-(1H-indol-3-yl)-2-methyl-2-[[(1S,3R,4S)-4,7,7-trimethyl-3-bicyclo[2.2.1]heptanyl]oxycarbonylamino]propanoyl]amino]-1-phenylethyl]amino]-4-oxobutanoic acid
CC1(C2CCC1(C(C2)OC(=O)NC(C)(CC3=CNC4=CC=CC=C43)C(=O)NCC(C5=CC=CC=C5)NC(=O)CCC(=O)O)C)C

Potent and selective CCK2 antagonist

Potent and selective, nonpeptide CCK 2 receptor antagonist (IC 50 values are 2.8 and 1232 nM for CCK 2 and CCK 1 respectively) that displays negligible affinity at GABA A benzodiazepine, substance P, neurotensin, opioid, bradykinin and 5-HT 3 receptors (IC 50 > 10 μM). Exhibits anxiolytic activity in elevated plus maze and social interaction tests and increases food intake in rats.
Quantity 50mg
Formula Weight 616.76
Percent Purity >98%
Chemical Name or Material PD 135158

Recommended Storage : Store at +4°C