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PG 01, Tocris Bioscience™

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Quantity:
10mg
50mg
This item is not returnable. View return policy
853138-65-5
C28H29N3O2
439.559
PQAYCXMQTUEDRD-UHFFFAOYSA-N
phenylglycine-01,2-2-1h-indol-3-yl-acetyl-methylamino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-yl-n-methylacetamido-n-4-isopropylphenyl-2-phenylacetamide,d03pgv,pg hplc,n-methyl-n-2-4-1-methylethyl phenyl amino-2-1h-indole-3-acetamide,2-1h-indol-3-ylacetyl methyl amino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-ylacetyl methylamino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-yl acetyl-methylamino-2-phenyl-n-4-propan-2-ylphenyl acetamide,2-2-1h-indol-3-yl-n-methylacetamido-2-phenyl-n-4-propan-2-yl phenyl acetamide
4695397
2-[[2-(1H-indol-3-yl)acetyl]-methylamino]-2-phenyl-N-(4-propan-2-ylphenyl)acetamide
CC(C)C1=CC=C(C=C1)NC(=O)C(C2=CC=CC=C2)N(C)C(=O)CC3=CNC4=CC=CC=C43
This item is not returnable. View return policy
853138-65-5
C28H29N3O2
439.559
PQAYCXMQTUEDRD-UHFFFAOYSA-N
phenylglycine-01,2-2-1h-indol-3-yl-acetyl-methylamino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-yl-n-methylacetamido-n-4-isopropylphenyl-2-phenylacetamide,d03pgv,pg hplc,n-methyl-n-2-4-1-methylethyl phenyl amino-2-1h-indole-3-acetamide,2-1h-indol-3-ylacetyl methyl amino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-ylacetyl methylamino-n-4-isopropylphenyl-2-phenylacetamide,2-2-1h-indol-3-yl acetyl-methylamino-2-phenyl-n-4-propan-2-ylphenyl acetamide,2-2-1h-indol-3-yl-n-methylacetamido-2-phenyl-n-4-propan-2-yl phenyl acetamide
4695397
2-[[2-(1H-indol-3-yl)acetyl]-methylamino]-2-phenyl-N-(4-propan-2-ylphenyl)acetamide
CC(C)C1=CC=C(C=C1)NC(=O)C(C2=CC=CC=C2)N(C)C(=O)CC3=CNC4=CC=CC=C43

CFTR potentiator; corrects F508del-CFTR conductance defect

Cystic fibrosis transmembrane conductance regulator (CFTR) potentiator. Corrects gating defects of CFTR mutants such as ΔF508 (Ka = 0.3 μM), E193K and G970R (Kd values are 0.22 μM and 0.45 μM respectively). Increases ΔF508-CFTR Cl- currents in the presence of forskolin; displays no effect on Ca2+-activated Cl- current.
Quantity 10mg
Formula Weight 439.55
Percent Purity >98%
Chemical Name or Material PG 01

Recommended Storage : Store at -20°C