Tocris™ PK-THPP

Potent TASK-3 channel blocker

Manufacturer: Tocris™ 5338/10

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Catalog No. 53-381-0

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For Research Use Only


    Description PK-THPP
    Quantity 10mg
    Product Type PK-THPP
    Molecular Weight 468.59
    Purity >99

    Potent TASK-3 channel blocker (IC50 = 35 and 300nM for TASK-3 and TASK-1 respectively). Increases breathing rate and induces respiratory alkalosis in rats.

    • Chemical Name: 1-[1-[6-[[1,1'-Biphenyl]-4-ylcarbonyl)-5,6,7,8-tetrahydropyrido[4,3-d]pyrimidin-4-yl]-4-piperidinyl]-1-butanone
    • Formula: C29H32N4O2
    • CAS Number: 1332454-07-5
    • Solubility: Soluble to 50mM in DMSO and to 20mM in 1eq. HCl with gentle warming
    • Purity: >99

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