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  8. PSB 11 hydrochloride, Tocris Bioscience™

PSB 11 hydrochloride, Tocris Bioscience™

Catalog Number p-4784365
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
453591-58-7
C16H18ClN5O
331.804
JAUSHKIWPLHBCN-RFVHGSKJSA-N
psb 11 hydrochloride, 8r-8-ethyl-1,4,7,8-tetrahydro-4-5h-imidazo 2,1-i purin-5-one hydrochloride, 8r-8-ethyl-4-methyl-2-phenyl-1,4,7,8-tetrahydro-5h-imidazo 2,1-i purin-5-one-hydrogen chloride 1/1
16759152
(8R)-8-ethyl-4-methyl-2-phenyl-7,8-dihydro-1H-imidazo[2,1-f]purin-5-one;hydrochloride
CCC1CN2C(=N1)C3=C(N=C(N3)C4=CC=CC=C4)N(C2=O)C.Cl
This item is not returnable. View return policy
453591-58-7
C16H18ClN5O
331.804
JAUSHKIWPLHBCN-RFVHGSKJSA-N
psb 11 hydrochloride, 8r-8-ethyl-1,4,7,8-tetrahydro-4-5h-imidazo 2,1-i purin-5-one hydrochloride, 8r-8-ethyl-4-methyl-2-phenyl-1,4,7,8-tetrahydro-5h-imidazo 2,1-i purin-5-one-hydrogen chloride 1/1
16759152
(8R)-8-ethyl-4-methyl-2-phenyl-7,8-dihydro-1H-imidazo[2,1-f]purin-5-one;hydrochloride
CCC1CN2C(=N1)C3=C(N=C(N3)C4=CC=CC=C4)N(C2=O)C.Cl

Description

Potent, selective hA3 receptor antagonist/inverse agonist

Potent and selective antagonist for the human adenosine A3 receptor, with low affinity for the rat A3 receptor (Ki values are 2.3 and > 10000 nM respectively). Displays > 1000-fold selectivity over human A1 and A2A receptors (Ki values are 4.1 and 3.3 μM respectively) and > 180-fold selectivity over rat A1, rat A2A and mouse A2B receptors. Acts as an inverse agonist in the [35S]GTPγS binding assay in hA3-CHO cells (IC50 = 36 nM).
Quantity 10 mg
Formula Weight 331.8
Percent Purity >98%
Chemical Name or Material PSB 11 hydrochloride

Safety and Handling

Recommended Storage Store at +4°C
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