Tocris™ R 1485 dihydrochloride

Selective and high affinity 5-HT6 antagonist

Manufacturer: Tocris™ 4964/10

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Catalog No. 49-641-0

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For Research Use Only


    Inhibitors R 1485 dihydrochloride
    Molecular Weight 450.35
    Product Type R 1485 dihydrochloride
    Purity >98
    Quantity 10mg

    Selective and high affinity 5-HT6 antagonist (pKi = 8.9); displays low hERG inhibition. Exhibits >100 fold selectivity against a panel of 50 targets including other 5-HT receptor subtypes. Brain penetrant.

    • Chemical Name: 4-[(2-Fluorophenyl)sulfonyl]-3,4-dihydro-8-(1-piperazinyl)-2H-1,4-benzoxazine dihydrochloride
    • Formula: C18H20FN3O3S.2HCl
    • Solubility: Soluble to 100mM in water and to 100mM in DMSO
    • Solubility: Soluble to 100mM in DMSO
    • Purity: >98

  • Description & Specifications

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