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SB 243213 dihydrochloride, Tocris Bioscience™

Catalog Number p-4817015
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Quantity:
10 mg
50 mg
This item is not returnable. View return policy
1780372-25-9
C22H21Cl2F3N4O2
501.331
UKMTYUXWLKQDNT-UHFFFAOYSA-N
sb 243213 dihydrochloride, 2,3-dihydro-5-methyl-n-6-2-methyl-3-pyridinyl oxy-3-pyridinyl-6-trifluoromethyl-1h-indole-1-carboxamide dihydrochloride
90488853
5-methyl-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide;dihydrochloride
CC1=C(C=C2C(=C1)CCN2C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C)C(F)(F)F.Cl.Cl
This item is not returnable. View return policy
1780372-25-9
C22H21Cl2F3N4O2
501.331
UKMTYUXWLKQDNT-UHFFFAOYSA-N
sb 243213 dihydrochloride, 2,3-dihydro-5-methyl-n-6-2-methyl-3-pyridinyl oxy-3-pyridinyl-6-trifluoromethyl-1h-indole-1-carboxamide dihydrochloride
90488853
5-methyl-N-[6-(2-methylpyridin-3-yl)oxypyridin-3-yl]-6-(trifluoromethyl)-2,3-dihydroindole-1-carboxamide;dihydrochloride
CC1=C(C=C2C(=C1)CCN2C(=O)NC3=CN=C(C=C3)OC4=C(N=CC=C4)C)C(F)(F)F.Cl.Cl

Selective 5-HT2C inverse agonist

Selective 5-HT2C inverse agonist (pKb = 9.8). Displays selectivity over other 5-HT2 subtypes (pKi values are 6.8, 7.0 and 9.0 for 5-HT2A, 5-HT2B and 5-HT2C respectively); also exhibits >100-fold selectivity over 50 other receptors, ion channels and enzymes. Displays anxiolytic activity in rat models.
Quantity 10 mg
Formula Weight 501.33
Percent Purity >99%
Chemical Name or Material SB 243213 dihydrochloride
Recommended Storage Store at +4°C
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