Potent and selective CB1 receptor antagonist (Ki = 7.8nM). Exhibits 1000-fold selectivity for CB1 over CB2 receptors. Inhibits CP 55,940-induced hypotension and WIN 55,212-2-induced hypothermia in vivo. Orally active.
Chemical Name: 3-(4-Chlorophenyl)-N-[(4-Chlorophenyl)sulfonyl]-4,5-dihydro-N'-methyl-4-phenyl-1H-pyrazole-1-carboximidamide
CAS Number: 362519-49-1
Solubility: Soluble to 100mM in DMSO and to 10mM in ethanol with gentle warming
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