Tocris™ SR 48692

Selective non-peptide NTS1 antagonist

Manufacturer: Tocris™ 3721/10

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Catalog No. 37-211-0R

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Disclaimers:

For Research Use Only


    Specifications

    Product Type SR 48692
    Inhibitors SR 48692
    Purity >98
    Molecular Weight 587.07
    Quantity 10mg

    Neurotensin antagonist; selective for NTS1 over NTS2 (apparent affinity, Ke, is 36nM for NTS1). Competitively inhibits binding of [125I]-neurotensin to HT29 and N1E115 cell membranes (IC50 values are 15.3 and 20.4nM respectively). Orally bioavailable.

    • Chemical Name: 2-[[[1-(7-Chloro-4-quinolinyl)-5-(2,6-dimethoxyphenyl)-1H-pyrazol-3-yl]carbonyl]amino]-tricyclo[3.3.1.13,7]decane-2-carboxylic acid
    • Formula: C32H31ClN4O5
    • CAS Number: 146362-70-1
    • Solubility: Soluble to 20mM in DMSO
    • Purity: >98

  • Description & Specifications

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