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SYM 2081, Tocris Bioscience™

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Quantity:
10mg
50mg
31137-74-3
C6H11NO4
161.157
KRKRAOXTGDJWNI-DMTCNVIQSA-N
2s,4r-4-methylglutamic acid,2s,4r-4-methylglutamate,2s,4r-2-amino-4-methylpentanedioic acid,4-methylglutamic acid,4-methylglutamate,4r-4-methyl-l-glutamic acid,threo-gamma-methylglutamate,2-amino-4-methyl-pentanedioic acid,tocris-0903,sym
95883
(2S,4R)-2-amino-4-methylpentanedioic acid
CC(CC(C(=O)O)N)C(=O)O
31137-74-3
C6H11NO4
161.157
KRKRAOXTGDJWNI-DMTCNVIQSA-N
2s,4r-4-methylglutamic acid,2s,4r-4-methylglutamate,2s,4r-2-amino-4-methylpentanedioic acid,4-methylglutamic acid,4-methylglutamate,4r-4-methyl-l-glutamic acid,threo-gamma-methylglutamate,2-amino-4-methyl-pentanedioic acid,tocris-0903,sym
95883
(2S,4R)-2-amino-4-methylpentanedioic acid
CC(CC(C(=O)O)N)C(=O)O

Highly selective kainate agonist

Potent and highly selective kainate receptor agonist, with an IC50 for inhibition of [3H]-kainate binding of 35 nM and almost 3,000- and 200-fold selectivity for kainate receptors over AMPA and NMDA receptors respectively. Also selectively inhibits the cloned excitatory amino acid transporter EAAT2 at higher concentrations. Also available as part of the Excitatory Amino Acid Transporter Inhibitor Tocriset™ and Kainate Receptor Tocriset™ .
Formula Weight 161.16
Percent Purity >97%
Quantity 50mg
Chemical Name or Material SYM 2081

Recommended Storage : Store at Room Temperature