Tocris™ TG 4-155

High affinity and selective EP2 receptor antagonist

Manufacturer: Tocris™ 5052/10

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Catalog No. 50-521-0

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For Research Use Only


    Product Type TG 4-155
    Inhibitors TG 4-155
    Purity >98
    Molecular Weight 394.46
    Quantity 10mg

    High affinity and selective EP2 receptor antagonist (KB values are 2.4 and 34.5nM for EP2 and DP1 receptors respectively). Exhibits >500-fold selectivity for EP2 over other prostanoid receptors. Inhibits butaprost-induced proinflammatory cytokine production, cell proliferation and invasion of PC-3 cells in vitro.

    • Chemical Name: (2E)-N-[2-(2-Methyl-1H-indol-1-yl)ethyl]-3-(3,4,5-trimethoxyphenyl)-2-propenamide
    • Formula: C23H26N2O4
    • CAS Number: 1164462-05-8
    • Solubility: Soluble to 100mM in DMSO and to 20mM in ethanol
    • Purity: >98

  • Description & Specifications

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