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Tocris Bioscience™ VU 0467485

Potent and selective positive allosteric modulator of M4 receptors; orally bioavailable and brain penetrant

$209.00 - $881.00

Specifications

CAS 1451994-10-7
Chemical Name or Material 5-Amino-N-[(3-fluoro-4-methoxyphenyl)methyl]-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide
Molecular Formula C17H17FN4O2S
Purity 98%
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Products 2
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
Catalog Number Mfr. No. Quantity Price Quantity & Availability  
69-321-0
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Tocris Bioscience™
6932/10
10 mg
Each for $209.00
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69-325-0
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Tocris Bioscience™
6932/50
50 mg
Each for $881.00
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Description

Description

  • Potent and selective positive allosteric modulator of M4 receptor; potentiates activity of ACh at M4 (EC50 values are 26.6 and 78.8 nM at rat and human M4 receptors, respectively).
  • Exhibits selectivity for M4 over human and rat M1-3, 5, and a panel of 200 other pharmacological targets.
  • Displays efficacy in a rat model of antipsychotic activity.
  • Orally bioavailable and brain penetrant.
Specifications

Specifications

1451994-10-7
5-Amino-N-[(3-fluoro-4-methoxyphenyl)methyl]-3,4-dimethylthieno[2,3-c]pyridazine-6-carboxamide
C17H17FN4O2S
98%
SDS
Product Certifications
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