Custom Enzymes and Inhibitors

Tocris Bioscience™ CHPG Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Selective mGlu5 agonist. Sodium salt of CHPG (Cat. No. 1049)

BD Caspase-9 Inhibitor, Z-LEHD-FMK Available on GSA/VA Contract for Federal Government customers only.

Irreversible and cell permeable inhibitor of caspase-9

Tocris Bioscience™ ATPγS Tetralithium Salt Available on GSA/VA Contract for Federal Government customers only.

P2 agonist; ATP (Cat. No. 3245) analog

Tocris Bioscience™ DL-AP5 Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Sodium salt of DL-AP5 (Cat. No. 0105)

Tocris Bioscience™ (5Z)-7-Oxozeaenol Available on GSA/VA Contract for Federal Government customers only.

Potent and selective TAK1 MAPKKK inhibitor

Tocris Bioscience™ AS 605240 Available on GSA/VA Contract for Federal Government customers only.

Potent and selective PI 3-kinase γ (PI 3-Kγ) inhibitor

Tocris Bioscience™ GSK 2606414

Potent and selective PERK inhibitor; orally bioavailable

Tocris Bioscience™ NSC 23766 Available on GSA/VA Contract for Federal Government customers only.

Selective inhibitor of Rac1-GEF interaction; antioncogenic

Tocris Bioscience™ Allopregnanolone Available on GSA/VA Contract for Federal Government customers only.

GABAA receptor positive allosteric modulator

Tocris Bioscience™ FR 180204 Available on GSA/VA Contract for Federal Government customers only.

Selective ERK inhibitor

Tocris Bioscience™ Teriflunomide

Dihydroorotate dehydrogenase inhibitor

Tocris Bioscience™ 2-MPPA Available on GSA/VA Contract for Federal Government customers only.

Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable

Tocris Bioscience™ Wnt-C59

Highly potent PORCN inhibitor

Tocris Bioscience™ Methylmalonate Available on GSA/VA Contract for Federal Government customers only.

Succinate dehydrogenase inhibitor

Tocris Bioscience™ MRS 2500 tetraammonium salt Available on GSA/VA Contract for Federal Government customers only.

Extremely potent and selective P2Y1 antagonist

Tocris Bioscience™ AbK Available on GSA/VA Contract for Federal Government customers only.

Photo-crosslinking probe

Tocris Bioscience™ Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor

Tocris Bioscience™ SID 26681509 Available on GSA/VA Contract for Federal Government customers only.

Cathepsin L inhibitor

Novus Biologicals™ TLR4 Inhibitor Peptide Set

Inhibits TLR4 signaling by blocking interactions between TLR4 and its adaptors Mal/TIRAP and TRAM

Tocris Bioscience™ Latrunculin A Available on GSA/VA Contract for Federal Government customers only.

Inhibitor of actin assembly and polymerization

Tocris Bioscience™ FRAX 486

Potent PAK inhibitor; brain penetrant and orally bioavailable

Tocris Bioscience™ ABT 702 dihydrochloride Available on GSA/VA Contract for Federal Government customers only.

Adenosine kinase inhibitor; orally active

Tocris Bioscience™ CP 376395 hydrochloride Available on GSA/VA Contract for Federal Government customers only.

Potent and selective CRF1 antagonist

Tocris Bioscience™ LY 379268 disodium salt Available on GSA/VA Contract for Federal Government customers only.

Sodium salt of LY 379268 (Cat. No. 2453); selective group II mGlu receptor agonist

R&D Systems™ proTAME Available on GSA/VA Contract for Federal Government customers only.

Cell-permeable APC/C inhibitor

Tocris Bioscience™ SB 328437 Available on GSA/VA Contract for Federal Government customers only.

Potent and selective CCR3 antagonist

Tocris Bioscience™ FIPI Available on GSA/VA Contract for Federal Government customers only.

Phospholipase D inhibitor

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