Custom Enzymes and Inhibitors

BD Caspase-9 Inhibitor, Z-LEHD-FMK Available on GSA/VA Contract for Federal Government customers only.

Irreversible and cell permeable inhibitor of caspase-9

Tocris Bioscience™ DL-AP5 Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Sodium salt of DL-AP5 (Cat. No. 0105)

Tocris Bioscience™ CHPG Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Selective mGlu5 agonist. Sodium salt of CHPG (Cat. No. 1049)

Tocris Bioscience™ Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor

Tocris Bioscience™ ATPγS Tetralithium Salt Available on GSA/VA Contract for Federal Government customers only.

P2 agonist; ATP (Cat. No. 3245) analog

Tocris Bioscience™ Teriflunomide

Dihydroorotate dehydrogenase inhibitor

Tocris Bioscience™ CP 376395 hydrochloride Available on GSA/VA Contract for Federal Government customers only.

Potent and selective CRF1 antagonist

Tocris Bioscience™ Wnt-C59

Highly potent PORCN inhibitor

Novus Biologicals™ MyD88 Inhibitor Peptide Set

For use in research applications

Tocris Bioscience™ LL 37

Antimicrobial peptide derivative of human cathelicidin

Tocris Bioscience™ Latrunculin A Available on GSA/VA Contract for Federal Government customers only.

Inhibitor of actin assembly and polymerization

BD General Caspase Inhibitor, Z-VAD-FMK Available on GSA/VA Contract for Federal Government customers only.

Cell permeable general caspase inhibitor that binds to the catalytic site of caspase proteases irreversibly and inhibits apoptosis

Tocris Bioscience™ 2-MPPA Available on GSA/VA Contract for Federal Government customers only.

Selective glutamate carboxypeptidase II (GCP II) inhibitor; orally bioavailable

Tocris Bioscience™ NSC 23766 Available on GSA/VA Contract for Federal Government customers only.

Selective inhibitor of Rac1-GEF interaction; antioncogenic

Tocris Bioscience™ NU 7441 Available on GSA/VA Contract for Federal Government customers only.

Potent and selective DNA-PK inhibitor

Novus Biologicals™ TLR4 Inhibitor Peptide Set

Inhibits TLR4 signaling by blocking interactions between TLR4 and its adaptors Mal/TIRAP and TRAM

Tocris Bioscience™ FR 180204 Available on GSA/VA Contract for Federal Government customers only.

Selective ERK inhibitor

Tocris Bioscience™ FRAX 486

Potent PAK inhibitor; brain penetrant and orally bioavailable

Tocris Bioscience™ GSK 2837808A Available on GSA/VA Contract for Federal Government customers only.

Potent, selective LDHA inhibitor

Tocris Bioscience™ Allopregnanolone Available on GSA/VA Contract for Federal Government customers only.

GABAA receptor positive allosteric modulator

Tocris Bioscience™ GSK 2606414

Potent and selective PERK inhibitor; orally bioavailable

Tocris Bioscience™ Tetrabenazine Available on GSA/VA Contract for Federal Government customers only.

Potent inhibitor of vesicular monoamine transport

Tocris Bioscience™ AR-C155858 Available on GSA/VA Contract for Federal Government customers only.

MCT1 and MCT2 inhibitor; inhibits glycolysis in cancer cells

BD FUT-175 (Futhan) Available on GSA/VA Contract for Federal Government customers only.

Synthetic, broad-specificity protease inhibitor and an inhibitor of the classical and alternate pathways of complement activation

Tocris Bioscience™ FIPI Available on GSA/VA Contract for Federal Government customers only.

Phospholipase D inhibitor

R&D Systems™ Boston Biochem Proteasome Inhibitor Z-Leu-Leu-Leu-CHO (MG-132)

Inhibits NF-kappaB activation. R&D Systems™ Boston Biochem Z-Leu-Leu-Leu-CHO (MG-132) is a proteasome and calpain inhibitor.

Tocris Bioscience™ MRS 2500 tetraammonium salt Available on GSA/VA Contract for Federal Government customers only.

Extremely potent and selective P2Y1 antagonist

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