Custom Enzymes and Inhibitors

Tocris Bioscience™ DL-AP5 Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Sodium salt of DL-AP5 (Cat. No. 0105)

Tocris Bioscience™ LL 37

Antimicrobial peptide derivative of human cathelicidin

Tocris Bioscience™ AbK Available on GSA/VA Contract for Federal Government customers only.

Photo-crosslinking probe

Tocris Bioscience™ CHPG Sodium salt Available on GSA/VA Contract for Federal Government customers only.

Selective mGlu5 agonist. Sodium salt of CHPG (Cat. No. 1049)

R&D Systems™ proTAME Available on GSA/VA Contract for Federal Government customers only.

Cell-permeable APC/C inhibitor

Tocris Bioscience™ Paroxetine maleate Available on GSA/VA Contract for Federal Government customers only.

Highly potent and selective 5-HT uptake inhibitor

Tocris Bioscience™ ATPγS Tetralithium Salt Available on GSA/VA Contract for Federal Government customers only.

P2 agonist; ATP (Cat. No. 3245) analog

Tocris Bioscience™ Wnt-C59

Highly potent PORCN inhibitor

Tocris Bioscience™ MRS 2500 tetraammonium salt Available on GSA/VA Contract for Federal Government customers only.

Extremely potent and selective P2Y1 antagonist

Tocris Bioscience™ W146 Available on GSA/VA Contract for Federal Government customers only.

Potent and selective S1P1 receptor antagonist

Tocris Bioscience™ PRT 4165

Inhibitor of Bmi1/Ring1A; blocks histone H2A ubiquitination

Tocris Bioscience™ Prostaglandin F2α

Naturally-occurring prostanoid; potent vasoconstrictor

Tocris Bioscience™ Tautomycetin

Selective PP1 inhibitor

BD FUT-175 (Futhan)

Synthetic, broad-specificity protease inhibitor and an inhibitor of the classical and alternate pathways of complement activation

Tocris Bioscience™ Aprotinin Available on GSA/VA Contract for Federal Government customers only.

Competitive serine protease inhibitor

Tocris Bioscience™ CP 376395 hydrochloride Available on GSA/VA Contract for Federal Government customers only.

Potent and selective CRF1 antagonist

Tocris Bioscience™ (5Z)-7-Oxozeaenol Available on GSA/VA Contract for Federal Government customers only.

Potent and selective TAK1 MAPKKK inhibitor

Tocris Bioscience™ LY 379268 disodium salt Available on GSA/VA Contract for Federal Government customers only.

Sodium salt of LY 379268 (Cat. No. 2453); selective group II mGlu receptor agonist

Tocris Bioscience™ MRS 2365 Available on GSA/VA Contract for Federal Government customers only.

Highly potent and selective P2Y1 agonist

Tocris Bioscience™ SB 204990 Available on GSA/VA Contract for Federal Government customers only.

ATP citrate lyase (ACLY) inhibitor

Tocris Bioscience™ a2-AdrenoceptorTocris Bioscience™et™

Selection of 5 α2-adrenoceptor ligands (Cat. Nos. 1030, 0425, 0928, 1133 and 0891)

Tocris Bioscience™ Tolvaptan

Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active

Tocris Bioscience™ E 64 Available on GSA/VA Contract for Federal Government customers only.

Potent and irreversible cysteine protease inhibitor

Tocris Bioscience™ KN 93 phosphate Available on GSA/VA Contract for Federal Government customers only.

CaM kinase II inhibitor; water soluble version of KN 93 (Cat. No. 1278).

Tocris Bioscience™ NU 7441 Available on GSA/VA Contract for Federal Government customers only.

Potent and selective DNA-PK inhibitor

Tocris Bioscience™ R 59-022

Diacylglycerol kinase inhibitor; increases PKC activity

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