Azolines
Medchemexpress LLC 1H-Benzimidazole, 2-(2-pyridinyl)- | 1137-68-4 | 99.9% | 195.22 | 100 G
2-(2'-Pyridyl)benzimidazole is a potentially tridentate ligand capable of forming stable complexes with various transition metal ions. It can function as an anti-inflammatory agent and an inhibitor of *Escherichia coli* methionine aminopeptidase.
- Potentially tridentate ligand
- Forms stable complexes with various transition metal ions
- Can be used as an anti-inflammatory agent
- Functions as an inhibitor of *Escherichia coli* methionine aminopeptidase
- For research use only
eMolecules 75-66-1 | 2-Methyl-2-propanethiol | Oakwood Chemicals | MFCD00004857 | 90.180 | C4H10S | 99.000 | CC(C)(C)S | 25g | 480148923
2-Methyl-2-propanethiol | Oakwood Chemicals | 75-66-1 | MFCD00004857 | 90.180 | C4H10S | 99.000 | CC(C)(C)S | 25g | 480148923
Medchemexpress LLC 1H-Benzimidazole, 2-(2-pyridinyl)- | 1137-68-4 | 99.9% | 195.22 | 10 G
2-(2′-Pyridyl)benzimidazole is a potentially tridentate ligand capable of forming stable complexes with various transition metal ions. It functions as an anti-inflammatory agent and effectively inhibits Escherichia coli methionine aminopeptidase, making it suitable for biochemical research. This compound appears as a solid, ranging from pale purple to purple or colorless to light pink and is intended for research use only.
- Functions as an anti-inflammatory agent
- Inhibits Escherichia coli methionine aminopeptidase
- IC50 of 13.3 μM in inhibiting human MetAP2 expressed in Sf9 cells
- Molecular formula: C12H9N3
- Molecular weight: 195.22
- Purity: 99.88%
- Ships at room temperature
- Stable for up to 3 years at room temperature
- Consistent with 1H NMR spectrum and LCMS
Medchemexpress LLC VH032 thiol | 2098836-54-3 | 95.9% | 490.64 | 1 ML
VH032 thiol (VHL ligand 6) is a VHL ligand. It binds to pan-BET inhibitor JQ1 via a linker to form PROTAC. VHL is a substrate recognition subunit of two ubiquitously expressed and biologically important Cullin RING E3 ubiquitin ligase complexes. It is also one of the most popular E3 ligases recruited by bifunctional Proteolysis-targeting chimeras (PROTACs) to induce ubiquitination and subsequent proteasomal degradation of a target protein.
- Binds to JQ1 to form PROTACs.
- Recruits VHL E3 ligase for protein degradation.
- Useful in the study of Proteolysis-targeting chimeras.
eMolecules 34301-54-7 | Adamantane-1-thiol | Accela ChemBio (ASD)168.300 | C10H16S | 98.000 | SC12CC3CC(CC(C3)C1)C2 | 5g | 485582438
Adamantane-1-thiol | Accela ChemBio (ASD) | 34301-54-7168.300 | C10H16S | 98.000 | SC12CC3CC(CC(C3)C1)C2 | 5g | 485582438
Medchemexpress LLC DOTA-thiol | 865470-67-3 | MFCD11501203 | 98.9% | 463.55 g/mol | C18H33N5O7S | 10 MG
DOTA-Thiol is a bifunctional chelator - a macrocyclic DOTA derivative - intended for tumor pre-targeting and for conjugation to peptides and radionuclides. It contains a thiol functional group that enables site-specific attachment and is supplied at high purity for research applications.
- Bifunctional chelator with a reactive thiol group
- Enables conjugation of peptides and radionuclides
- Suitable for tumor pre-targeting and radiolabeling workflows
- High purity for research-grade use
- Available in milligram-scale pack sizes for synthesis and labeling
![Medchemexpress LLC M-PEG-thiol (MW 2000) | 134874-49-0 | 99.8% | COCCOCCS.[MW 2000].[n] | 1 G](https://assets.fishersci.com/TFS-Assets/CCG/product-images/default.jpg-250.jpg)
Medchemexpress LLC M-PEG-thiol (MW 2000) | 134874-49-0 | 99.8% | COCCOCCS.[MW 2000].[n] | 1 G
m-PEG-thiol (MW 2000) is a PEG-based PROTAC linker used in the synthesis of PROTACs. This product is intended for research use only.
- PEG-based PROTAC linker
- Used in the synthesis of PROTACs
- Exploits the intracellular ubiquitin-proteasome system
- Selectively degrades target proteins
Medchemexpress LLC Methimazole-d3 | 1160932-07-9 | 99.7% | 1 MG
Methimazole-d3 is a deuterium labeled anti-thyroid agent, derived from Methimazole (Thiamazole), which blocks thyroid hormone production. Deuteration can impact the pharmacokinetic and metabolic profiles of drugs. This compound is for research use only.
- Can be used as a tracer
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS
Medchemexpress LLC NAG-thiazoline | 179030-22-9 | ≥95.0% | 219.26 | 50 MG
NAG-thiazoline is an O-GlcNAcase inhibitor with a Ki of 180 nM. It is also a potent GH20 GlcNAcase (VhGlcNAcase) inhibitor with an IC50 of 11.9 μM and a Ki of 62 μM.
- Completely inhibits the growth of V. campbellii strain 650 with a MIC value of 0.5 μM.
- O-GlcNAcase inhibitor.
- Potent GH20 GlcNAcase (VhGlcNAcase) inhibitor.
Accela Chembio Inc 2-amino-5-bromothiazole | 5g | 3034-22-8 | MFCD00016893 | 95+% | Shelf Life: 1080 Days | Light Sensitive/nitrogen Or Argon/-20
2-amino-5-bromothiazole | 5g | 3034-22-8 | MFCD00016893 | 95+% | Shelf Life: 1080 Days | Light Sensitive/nitrogen Or Argon/-20
Medchemexpress LLC 2-methyl-2-thiazoline-4-carboxylic acid, sodium | 15058-19-2 | MFCD03093520 | 98.1% | 167.16 | C5H6NNaO2S | 250 MG
2-Methyl-2-thiazoline-4-carboxylic acid sodium is the sodium salt of a thiazoline-class heterocycle supplied as a research-grade solid reagent. It is intended for laboratory research and analytical applications where a well-characterized heterocyclic building block is required; not for human or clinical use.
- Sodium salt form for improved solubility in aqueous media.
- High reported purity of 98.1%.
- Molecular formula C5H6NNaO2S and molecular weight 167.16 g/mol.
- Supplied in small pack sizes suitable for research-scale use.
- Suitable as a reagent or building block in organic synthesis and analytical workflows.
Medchemexpress LLC NAG-thiazoline | 179030-22-9 | ≥95.0% | 219.26 | 25 MG
NAG-thiazoline is an O-GlcNAcase inhibitor with a Kᵢ of 180 nM. It is also a potent GH20 GlcNAcase (VhGlcNAcase) inhibitor with an IC₅₀ of 11.9 μM and a Kᵢ of 62 μM. It completely inhibits the growth of V. campbellii strain 650. This product is for research use only.
- O-GlcNAcase inhibitor (Kᵢ of 180 nM)
- Potent GH20 GlcNAcase (VhGlcNAcase) inhibitor (IC₅₀ of 11.9 μM, Kᵢ of 62 μM)
- Inhibits the growth of V. campbellii strain 650 (MIC value of 0.5 μM)
- Suitable for research applications
