Azoles
![Medchemexpress LLC 6-bromo-7-[4-[(5-methyl-3-isoxazolyl)methyl]-1-piperazinyl]-2-[4-(4-methyl-1-piperazinyl)phenyl] | 1095382-05-0 | ≥98.0% | 551.48 g·mol⁻¹ | C26H31BrN8O | 5 MG](https://assets.fishersci.com/TFS-Assets/CCG/product-images/VN00132390-HY-10804-5MG.JPG-250.jpg)
Medchemexpress LLC 6-bromo-7-[4-[(5-methyl-3-isoxazolyl)methyl]-1-piperazinyl]-2-[4-(4-methyl-1-piperazinyl)phenyl] | 1095382-05-0 | ≥98.0% | 551.48 g·mol⁻¹ | C26H31BrN8O | 5 MG
A potent, orally available Aurora kinase inhibitor active against Aurora A, B, and C that displays antiproliferative activity in multiple tumor cell lines. The compound is supplied as a powder for research use and has documented solubility and storage recommendations for both powder and solution forms.
- Potent inhibition of Aurora A, B, and C with IC50s of 15, 25, and 19 nM.
- Orally bioavailable compound showing antiproliferative activity in tumor cell lines.
- Supplied as a powder with high purity (≥98% by HPLC).
- Molecular weight 551.48 g·mol⁻¹ and formula C26H31BrN8O.
- Soluble in DMSO (16.67 mg/mL) and compatible with common vehicle formulations.
- Recommended storage: powder at -20°C (3 years) or 4°C (2 years); in solvent at -80°C (2 years).
Medchemexpress LLC HY-111503 10mg Medchemexpress, Y06137 CAS:2226534-49-0 Purity:>98%
Medchemexpress, HY-111503 10mg Y06137 CAS:2226534-49-0 Y06137 is a potent and selective BET inhibitor for treatment of castration-resistant prostate cancer (CRPC). Y06137 binds to the BRD4(1) bromodomain with a Kd of 81 nM. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-10505 5mg Medchemexpress, Orteronel CAS:566939-85-3 Purity:>98%
Medchemexpress, HY-10505 5mg Orteronel CAS:566939-85-3 Orteronel is a highly selective inhibitor of human 17,20-lyase with IC50 of 38 nM, and exhibits >1000-fold selectivity over other CYPs such as 11-hydroxylase and CYP3A4. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-103186 10mg Medchemexpress, MRS-1706 CAS:264622-53-9 Purity:>98%
Medchemexpress, HY-103186 10mg MRS-1706 CAS:264622-53-9 MRS-1706 is a potent and selective adenosine A2B receptor inverse agonist. MRS-1706 has Ki values of 1.39, 112, 157, and 230 nM for human A2B, A2A, A1 and A3 receptors respectively. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC 2-phenylimidazole | 670-96-2 | 99.2% | 144.18 | C9H8N2 | 500g
2-Phenylimidazole (PhI) is a corrosion inhibitor for brass and can be used to prepare complexes with ruthenium (III)[1]
Medchemexpress LLC HY-108939 1mg Medchemexpress, Aminoacyl tRNA synthetase-IN-1 CAS:219931-45-0 Purity:>98%
Medchemexpress, HY-108939 1mg Aminoacyl tRNA synthetase-IN-1 CAS:219931-45-0 Aminoacyl tRNA synthetase-IN-1 is a bacterial aminoacyl tRNA synthetase (aaRS) inhibitor. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-108900 1mg Medchemexpress, Leu-AMS CAS:288591-93-5 Purity:>98%
Medchemexpress, HY-108900 1mg Leu-AMS CAS:288591-93-5 Leu-AMS (compound 6), a leucine analogue, is a potent inhibitor of leucyl-tRNA synthetase (LRS) with an IC50 of 22.34 nM, which inhibits the catalytic activity of LRS but did not affect the leucine-induced mTORC1 activation. Leu-AMS shows cytotoxicity in cancer cells and normal cells, and inhibits the growth of bacteria. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC HY-103181 50mg Medchemexpress, N6-Cyclopentyladenosine CAS:41552-82-3 Purity:>98%
Medchemexpress, HY-103181 50mg N6-Cyclopentyladenosine CAS:41552-82-3 N6-Cyclopentyladenosine (CPA) is a selective Adenosine A1 receptor agonist, with Ki values of 2.3 nM, 790 nM and 43 nM for human A1, A2A and A3 receptors, respectively. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Medchemexpress LLC TEAD3 Human His-SU 5ug
Recombinant human TEAD3 protein (residues M112-D435) with an N-terminal 6xHis-SUMO fusion tag, supplied as a small-scale purified protein for research applications.
- Contains residues M112-D435 of human TEAD3.
- N-terminal 6xHis-SUMO tag for affinity purification.
- Approximate molecular weight 52.3 kDa.
- Purity ~90% suitable for biochemical assays.
- Provided in a 5 μg size for small-scale experiments.
Medchemexpress LLC HY-104021 10mg Medchemexpress, GSK840 CAS:2361146-30-5 Purity:>98%
Medchemexpress, HY-104021 10mg GSK840 CAS:2361146-30-5 GSK840 (GSK'840) is a receptor-interacting protein kinase 3 (RIP3 or RIPK3) inhibitor, which binds RIP3 kinase domain with an IC50 of 0.9 nM, and inhibits kinase activity with an IC50 of 0.3 nM. Purity:>98% Medchemexpress has over 10000 novel life-science reagents, reference compounds, APIs and natural compounds for laboratory and scientific use. Other quantity can also be offered.
Chem-Impex International, Inc. Isoxazole | 288-14-2 | MFCD00003149 | 25G
Isoxazole, 288-14-2, MFCD00003149, 25G
Matrix Scientific 2-BROMO-5-METHYLTHIAZOLE2-BR-5
2-bromo-5-methylthiazole Mf C4h4brns Mw 178.06 Cas 41731-23-1 Mdl MFCD08460610
Sigma Aldrich Fine Chemicals Biosciences 1,3-Di-tert-butylimidazolium tetrafluoroborate 97% | 263163-17-3 | MFCD07784425 | 1G
1,3-Di-tert-butylimidazolium tetrafluoroborate 97% | Purity: 97% | Mol Wt: 268.1 | 263163-17-3 | MFCD07784425 | 1G
