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Medchemexpress LLC 1-[4-[(5-cyclopropyl-1H-pyrazol-3-yl)amino]pyrrolo[2,1-f]triazin-2-yl]-N-(6-fluoro-3-p... | 1001350-96-4 | MFCD18633202 | 99.4% | 461.5 g/mol | C23H24FN9O | 25 MG

Supplier: Medchemexpress LLC HY1020025MG
BMS-754807 is a potent, reversible small-molecule inhibitor of the insulin-like growth factor 1 receptor (IGF-1R) and the insulin receptor (InsR) used in oncology and signal-transduction research. It shows low-nanomolar activity against several kinases and is supplied at high purity for in vitro and in vivo studies.
- Potent IGF-1R and InsR inhibition (IC50 ~1.7-1.8 nM).
- Binding affinity Ki <2 nM.
- Additional kinase activity against Met, RON, TrkA, TrkB, AurA, and AurB.
- High purity (99.42%).
- CAS number 1001350-96-4 for unambiguous identification.
- Chemical formula C23H24FN9O; molecular weight 461.5 g/mol.
- Available in small milligram quantities, including 25 MG packs for research use.
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