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Medchemexpress LLC 2-(3,5-difluoro-4-hydroxyphenylamino)-8-isopentyl-5,7-dimethyl-7,8-dihydropteridin-6(5H)-one | 501437-28-1 | MFCD11223662 | >98.0% | 391.42 g·mol⁻¹ | C19H23F2N5O2 | 500 MG
SDP

Supplier:  Medchemexpress LLC HY10510500MG

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BI-D1870 is a potent, ATP-competitive inhibitor of the p90 ribosomal S6 kinase (RSK) family. It is cell permeable and reported to penetrate the brain, making it suitable for cellular and in vivo studies of RSK-mediated signaling and related biological processes.

  • Selective ATP-competitive inhibitor of RSK isoforms.
  • Low nanomolar potency against RSK1-RSK4 (IC50s: 31, 24, 18, 15 nM).
  • Cell permeable for use in cellular assays.
  • Reported brain penetration supports in vivo applications.
  • Useful for studying MAPK/ERK-RSK signaling pathways.
  • Available as a solid suitable for storage and formulation.

Catalog No. 50-002-43557


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