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Medchemexpress LLC 2-pyrazinecarboxamide, 6-ethyl-5-[(trans-4-methoxycyclohexyl)amino] | 1373409-08-5 | 98.0% | 580.76 g/mol | C31H48N8O3 | 5 MG
SDP

Supplier:  Medchemexpress LLC HY1117525MG

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EML4-ALK kinase inhibitor 1 is a potent, orally active small-molecule inhibitor of the EML4-ALK fusion kinase. Reported biochemical potency is IC50 = 1 nM, and the compound shows cellular antiproliferative activity in BaF3 cells expressing EML4-ALK. Supplied as a high-purity research reagent for in vitro and in vivo studies.

  • Potent biochemical inhibition (IC50 1 nM).
  • Demonstrated antiproliferative activity in EML4-ALK BaF3 cells (~9.7 nM).
  • High purity 98.0%.
  • Molecular weight 580.76 g/mol; formula C31H48N8O3.
  • Soluble in DMSO (110 mg/mL) and compatible with reported in vivo formulations.
  • Available in milligram pack sizes for research use.

Catalog No. 50-002-63307


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