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Medchemexpress LLC (4R)-1,3,4,5-tetrahydro-4-methyl-6-[1-methyl-3-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-5-yl]-2H-1,5-be | 1884712-47-3 | MFCD30489741 | 99.9% | 386.45 | C22H22N6O | 50 MG
SDP

Supplier:  Medchemexpress LLC HY10048250MG

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CPI-637 is a selective, cell-active benzodiazepinone inhibitor of the CBP and EP300 bromodomains used as a research reagent for epigenetic and cancer-biology studies. It shows nanomolar biochemical potency and cellular target engagement and is supplied as a high-purity solid for laboratory use.

  • Selective CBP/EP300 bromodomain inhibition (CBP IC50 ≈ 0.03 μM; EP300 IC50 ≈ 0.051 μM).
  • Low activity against BRD4 BD-1 (IC50 ≈ 11.0 μM), indicating >700-fold selectivity.
  • Cellular activity with CBP BRET EC50 ≈ 0.3 μM.
  • High purity solid suitable for biochemical and cellular assays.
  • Stable under recommended storage conditions (powder: -20°C; in solvent: -80°C).
  • Available in small research package sizes (for example, 50 mg).

Catalog No. 50-002-13781


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