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Medchemexpress LLC ASP-9521 | 1126084-37-4 | 98.0% | 330.42 | 100 MG
Supplier: Medchemexpress LLC HY19903100MG
ASP-9521 is a potent, selective, and orally available AKR1C3 inhibitor with an IC50 of 11 nM for human AKR1C3, intended for research use only.
- Potent, selective, and orally available AKR1C3 inhibitor.
- IC50 of 11 nM for human AKR1C3 and 49 nM for monkey AKR1C3.
- Shows more than 100-fold selectivity for AKR1C3 over the isoform AKR1C2.
- Suppresses AD-dependent PSA production and cell proliferation in cells.
- Inhibits AD-induced intratumoural T production in xenografts.
- Bioavailability after oral administration is 35% in rats, 78% in dogs, and 58% in monkeys.
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