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Medchemexpress LLC Benzenesulfonamide, N-[2-[(1-amino-6-isoquinolinyl)oxy]-4-methylphenyl]-2-methoxy- | 2377379-39-8 | 99.9% | 435.50 | 5 MG
SDP

Supplier:  Medchemexpress LLC 5MGHY130118

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MRGPRX1 agonist 1 is a highly potent MRGPRX1 agonist (EC₅₀=50 nM) with greater than 50-fold selectivity for δ, μ, and κ opioid receptors. It is inactive against MRGPRC11, which inhibits high voltage-activated Ca²⁺ currents and mitigates nociceptive transmission. This compound is useful for studying chronic pain, especially neuropathic pain.

  • Highly potent MRGPRX1 agonist (EC₅₀=50 nM)
  • Demonstrates greater than 50-fold selectivity for δ, μ, and κ opioid receptors
  • Inactive against MRGPRC11
  • Useful for studying chronic pain, particularly neuropathic pain
  • Soluble in DMSO at 125 mg/mL
  • Powder stable at -20°C for 3 years, 4°C for 2 years
  • In solvent stable at -80°C for 6 months, -20°C for 1 month

Catalog No. 50-003-64630


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