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Medchemexpress LLC BI-3663 | 2341740-84-7 | 99.8% | 917.84 | 1 MG
SDP

Supplier:  Medchemexpress LLC HY11154610MM/1ML

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BI-3663 is a highly selective PTK2/FAK PROTAC that utilizes Cereblon ligands to hijack E3 ligases for PTK2 degradation. It inhibits PTK2 with an IC50 of 18 nM and demonstrates anti-cancer activity. It potently degrades PTK2 in Hep3B2.1-7 cells and A549 cells, with pDC50s of 7.6 and 7.9, respectively.

  • Highly selective PTK2/FAK PROTAC
  • Utilizes Cereblon ligands for PTK2 degradation
  • Inhibits PTK2 with an IC50 of 18 nM
  • Demonstrates anti-cancer activity
  • Potently degrades PTK2 in Hep3B2.1-7 cells and A549 cells

Catalog No. 50-003-47154


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