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Cayman Chemical BIsoprololhemIfumarate 100mg
SDP

Supplier:  Cayman Chemical 23827100 MG

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A β1-AR antagonist (Ki = 25 nM for the human receptor); selective for β1- over β2-ARs (Ki = 480 nM for the human receptor in a radioligand binding assay); binds to rat ventricular myocytes and heart membranes that endogenously express β1-ARs and β1- and β2-ARs, respectively (Kis = 20 and 38.1 nM, respectively); inhibits isoproterenol-induced increases in heart rate and myocardial contractility in conscious dogs at 0.3 mg/kg; decreases blood pressure and heart rate in SHRs at 7.5 mg/kg twice per day over 19 weeks; inhibits SARS-CoV-2 Mpro (IC50 = 118.5 UG/ml) and reduces viral infectivity in SARS-CoV-2 infected Vero E6 cells (IC50 = 15.917 UG/ml)

Catalog No. 50-299-4807


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