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Medchemexpress LLC Brilanestrant | 1365888-06-7 | 99.9% | 100 MG

Supplier: Medchemexpress LLC HY12864100MG
Brilanestrant is an orally bioavailable selective estrogen receptor degrader (SERD) with an IC50 of 0.7 nM. It is intended for research use only.
- Orally bioavailable selective estrogen receptor degrader
- Potent ER-α binder
- Full transcriptional antagonist with no agonism
- Induces ER-α degradation
- Shows efficacy in MCF-7 breast cancer cell viability assays
- Exhibits low clearance and good oral bioavailability
- Demonstrates tumor-growth inhibition in MCF-7 xenograft models
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