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Medchemexpress LLC BSJ-03-204 | 2349356-09-6 | 99.8% | 832.90 | 1 MG
Supplier: Medchemexpress LLC HY1362501MG
BSJ-03-204 is a PROTAC connected by ligands for Cereblon and CDK. It is a potent and selective Palbociclib-based CDK4/6 dual degrader (PROTAC), with IC50s of 26.9 nM for CDK4/D1 and 10.4 nM for CDK6/D1. BSJ-03-204 does not induce IKZF1/3 degradation and exhibits anti-cancer activity.
- Potent anti-proliferative effects on MCL cell lines.
- Potently induces a G1 arrest.
- Selectively degrades CDK4/6 in WT cells, not IKZF1/3.
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