Learn More
TARGETMOL CHEMICALS INC CF53 5MG

Supplier: TARGETMOL CHEMICALS INC T107735MG
Also available in 1 mg 10 mg 25 mg 50 mg 100 mg 1 mL 10 mM (in DMSO) and bulk. Please contact Fisher for quotes. CF53 is a highly potent selective and orally active inhibitor of BET protein with a Ki of <1 nM Kd of 2.2 nM and an IC50 of 2 nM for BRD4 BD1. CF53 binds to both the BD1 and BD2 domains of BRD2 BRD3 BRD4 and BRDT BET proteins with high affinities very selective over non-BET bromodomain-containing proteins. CF53 shows potent anti-tumor activity both in vitro and in vivo. purity: 100%
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.