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Selleck Chemical LLC Enitociclib S8730-100MG
Supplier: Selleck Chemical LLC S8730100MG
Enitociclib (BAY 1251152) is a potent PTEFb/CDK9 inhibitor with an IC50 value of 3 nM for CDK9 and an at least 50-fold selectivity against other CDKs in enzymatic assays BAY1251152 binds to and blocks the phosphorylation and kinase activity of CDK9 thereby preventing PTEFb-mediated activation of RNA Pol II and leading to the inhibition of gene transcription of various anti-apoptotic proteins
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