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Medchemexpress LLC Fulvestrant-d3 (ICI 182780-d3) | 129453-61-8 | 97.6% | 609.79 | 1 MG
Supplier: Medchemexpress LLC HY13636S1MG
Fulvestrant-d3 is a deuterium-labeled form of Fulvestrant (ICI 182780). Fulvestrant is a potent estrogen receptor (ER) antagonist with an IC50 of 9.4 nM and a pure antiestrogen. It acts as a GPR30 agonist and effectively inhibits the growth of ER-positive MCF-7 cells with an IC50 of 0.29 nM. Additionally, Fulvestrant induces autophagy and exhibits antitumor efficacy. This compound is intended for research use, specifically as a tracer and an internal standard for quantitative analysis methods like NMR, GC-MS, or LC-MS.
- Deuterium labeled Fulvestrant.
- Can be used as a tracer.
- Can be used as an internal standard for quantitative analysis by NMR, GC-MS, or LC-MS.
- Stable heavy isotopes are incorporated for quantitation during drug development.
- Deuteration can potentially affect the pharmacokinetic and metabolic profiles of drugs.
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