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Medchemexpress LLC Gabapentin enacarbil | 478296-72-9 | 95.0% | 329.39 | 1 ML

Supplier: Medchemexpress LLC HY1621610MM/1ML
Gabapentin enacarbil (XP-13512) is a prodrug of Gabapentin designed for absorption throughout the intestine by high-capacity nutrient transporters. Gabapentin is an orally active P/Q type Ca2+ channel blocker. This product can be used for the study of Restless Legs Syndrome (RLS) and postherpetic neuralgia (PHN).
- Prodrug of gabapentin.
- Absorbed throughout the intestine by high-capacity nutrient transporters.
- Used for the study of restless legs syndrome (RLS) and postherpetic neuralgia (PHN).
- Stable at physiological pH.
- Rapidly converted to gabapentin in intestinal and liver tissue from rats, dogs, monkeys, and humans.
- Improved oral bioavailability, dose proportionality, and enhanced colonic absorption compared with gabapentin in rats and monkeys.
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