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Medchemexpress LLC GAK inhibitor 49 | 319492-82-5 | MFCD29701419 | 98.8% | 370.40 g·mol-1 | C20H22N2O5 | 10MG
Supplier: Medchemexpress LLC HY12479310MG
GAK inhibitor 49 is a potent, ATP-competitive, and highly selective inhibitor of cyclin G-associated kinase (GAK) developed for research applications. It exhibits sub-nanomolar biochemical potency (Ki = 0.54 nM) and cellular activity (cell IC50 ≈ 56 nM). The compound has formula C20H22N2O5 and a molecular weight of 370.40 g·mol-1. It is typically supplied in small research quantities and is reported with high purity (reported values ≈98.8% to ≥99%).
- Potent ATP-competitive GAK inhibitor (Ki = 0.54 nM).
- Demonstrates cellular activity (cell IC50 ≈ 56 nM).
- High selectivity with limited off-target binding reported.
- Suitable for in vitro biochemical and cell-based assays.
- Supplied in research-scale quantities for screening and profiling.
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