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Medchemexpress LLC GNE-272 | 1936428-93-1 | MFCD30738051 | 99.6% | 424.47 g·mol⁻¹ | C22H25FN6O2 | 100 MG
SDP

Supplier:  Medchemexpress LLC HY100726100MG

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GNE-272 is a potent, selective small-molecule probe that targets the bromodomains of CBP and EP300. It exhibits low-nanomolar biochemical potency and shows cellular activity including inhibition of MYC expression, making it suitable for in vitro and in vivo probe studies when handled as a research-grade compound.

  • Potent CBP/EP300 bromodomain inhibition (CBP IC50 0.02 μM, EP300 IC50 0.03 μM).
  • Lower affinity for BRD4 (IC50 13 μM).
  • Demonstrated cellular activity (MV4-11 MYC inhibition EC50 1.9 μM).
  • High reported purity (99.6%).
  • Supplied as powder and as DMSO solution for ready reconstitution.
  • Storage stability data provided for powder and solvent forms.

Catalog No. 50-002-14417


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