Learn More
Medchemexpress LLC GSK-5959 | 901245-65-6 | 99.7% | 394.47 | 50 MG

Supplier: Medchemexpress LLC HY1866550MG
GSK-5959 is a potent, selective, and cell-permeable BRPF1 bromodomain inhibitor. It is intended for research use only and not sold to patients.
- Potent, selective, and cell permeable BRPF1 bromodomain inhibitor.
- Displays selectivity over BRPF2 (100-fold) and BRPF3 (>1000-fold).
- Exhibits an EC50 = 0.98 μM in cellular NanoBRET assay.
- Has no effect on TRIM24 SUMOylation.
By clicking Submit, you acknowledge that you may be contacted by Fisher Scientific in regards to the feedback you have provided in this form. We will not share your information for any other purposes. All contact information provided shall also be maintained in accordance with our Privacy Policy.