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Medchemexpress LLC GSK256066 trifluoroacetate | 1415560-64-3 | 99.8% | 632.61 g·mol⁻¹ | C29H27F3N4O7S | 10 MG
SDP

Supplier:  Medchemexpress LLC HY7006910MG

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The trifluoroacetate salt of GSK256066 is a selective, high-affinity phosphodiesterase 4 (PDE4) inhibitor used in preclinical research on respiratory inflammatory diseases such as COPD. It displays picomolar potency against PDE4B and suppresses LPS-induced tumor necrosis factor α production in human monocytes.

  • High affinity for PDE4B (IC50 ≈ 3.2 pM)
  • Inhibits LPS-stimulated TNFα production (IC50 ≈ 0.01 nM)
  • High selectivity versus other PDE families
  • Supplied as a trifluoroacetate salt for improved handling
  • Available in small research pack sizes suitable for assay development

Catalog No. 50-002-98636


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