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Medchemexpress LLC Icotinib (Hydrochloride) | 1204313-51-8 | C22H22ClN3O4 | 100 MG
Supplier: Medchemexpress LLC HY15164100MG
Icotinib Hydrochloride (BPI-2009) is a potent, CNS-penetrant, and specific EGFR inhibitor with an IC50 of 5 nM. It inhibits mutant EGFRL858R, EGFRL858R/T790M, EGFRT790M, and EGFRL861Q. This compound is a click chemistry reagent containing an Alkyne group, enabling it to undergo copper-catalyzed azide-alkyne cycloaddition (CuAAc) with molecules containing Azide groups.
- Potent, CNS-penetrant, and specific EGFR inhibitor
- Inhibits mutant EGFRL858R, EGFRL858R/T790M, EGFRT790M, and EGFRL861Q
- Click chemistry reagent for copper-catalyzed azide-alkyne cycloaddition
- Exhibits potent dose-dependent antitumor effects in nude mice
- Well tolerated at doses up to 120 mg/kg/day in mice
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