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Medchemexpress LLC Imlunestrant | 2408840-26-4 | 100.0% | C29H24F4N2O3 | 250 MG
Supplier: Medchemexpress LLC 250MGHY145572
Imlunestrant is an orally active, potent, and selective estrogen receptor degrader (SERD) with pure antagonistic properties. It leads to sustained inhibition of ER-dependent gene transcription and cell growth, making it suitable for research on ER-positive (ER+) advanced breast cancer (aBC) and endometrial endometrioid cancer (EEC).
- Orally active, potent, and selective estrogen receptor degrader (SERD)
- Pure antagonistic properties
- Sustained inhibition of ER-dependent gene transcription and cell growth
- Antiproliferative activity against human MCF7 cells harboring ERalpha Y537N mutant
- Antiproliferative activity against human MCF7 cells harboring wild type ERalpha
- Favorable pharmacokinetic (PK) properties
- Demonstrates antitumor activity in ESR1 mutants
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