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Medchemexpress LLC Opiranserin hydrochloride | 1440796-75-7 | 99.6% | 430.97 | 25 MG
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Supplier:  Medchemexpress LLC 25MGHY109067A

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Opiranserin hydrochloride is a non-opioid and non-NSAID analgesic candidate. It acts as a dual antagonist of glycine transporter type 2 (GlyT2) and serotonin receptor 2A (5HT2A). It also exhibits antagonistic activity on rP2X3. This compound is being developed as an injectable agent for the treatment of postoperative pain. In preclinical studies, it effectively reduced mechanical allodynia and pain-related behaviors, with efficacy comparable to morphine. It also reduced mechanical allodynia in a rat spinal nerve ligation model.

  • Acts as a dual antagonist of glycine transporter type 2 (GlyT2)
  • Antagonizes serotonin receptor 2A (5HT2A)
  • Exhibits antagonistic activity on rP2X3
  • Developed as an injectable agent for postoperative pain
  • Effectively reduced mechanical allodynia and pain-related behaviors in preclinical studies

Catalog No. 50-003-47448


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