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Medchemexpress LLC PROTAC EZH2 Degrader-1 | 2641601-67-2 | 99.4% | 942.15 | 5 MG
SDP

Supplier:  Medchemexpress LLC HY1475255MG

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PROTAC EZH2 Degrader-1, also known as Compound 150d, is a potent PROTAC EZH2 Degrader. It exhibits an inhibitory effect on EZH2 methyltransferase activity with an IC50 of 2.7 nM. EZH2 is a crucial factor in the initiation and progression of various tumors. This product is intended for research use only.

  • Potent inhibition of EZH2 methyltransferase activity with an IC50 of 2.7 nM.
  • Demonstrates anti-proliferative activity against several cell lines including EOL1, MV4-11, Pfeiffer, RS4-11, and WSUDLCL2.
  • Enhances the sensitivity of H128-LM cells to Carboplatin, VP16, and VM26.
  • Exhibits antitumor activity in H128-LM xenograft mouse models, prolonging survival when combined with other agents.
  • High purity of 99.4%.

Catalog No. 50-003-60504


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