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Medchemexpress LLC Pyrrolo[3,4-b]pyrrole-5(1H)-carboxamide, N-[4-(3-ethynylphenyl)amino-7-methoxy-6-quinazolinyl]hex... | 1353644-70-8 | MFCD00038264 | 99.7% | 442.51 g/mol | C25H26N6O2 | 100 MG

Supplier: Medchemexpress LLC HY104066100MG
Theliatinib is a potent, ATP-competitive, orally active, and highly selective epidermal growth factor receptor (EGFR) inhibitor provided for research use. It shows low nanomolar cellular activity against EGFR and has been evaluated in preclinical models of EGFR-driven cancers.
- Potent EGFR inhibition (Ki ≈ 0.05 nM; IC50 ≈ 3 nM).
- Highly selective for EGFR over common off-target kinases.
- Suitable for in vitro and in vivo preclinical studies.
- High reported purity for reliable assay results.
- Formulation as a solid; soluble in DMSO for assay preparation.
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