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Medchemexpress LLC (Rac)-5-Hydroxymethyl Tolterodine hydrochloride | 250214-40-5 | C22H32ClNO2 | 500 MG
Supplier: Medchemexpress LLC HY76570A500MG
(Rac)-5-Hydroxymethyl Tolterodine hydrochloride is an active metabolite of Tolterodine, functioning as a muscarinic acetylcholine receptor (mAChR) antagonist. It exhibits Ki values of 2.3 nM, 2 nM, 2.5 nM, 2.8 nM, and 2.9 nM for M1, M2, M3, M4, and M5 receptors, respectively. This compound is suitable for research related to overactive bladder, demonstrating competitive inhibition of carbachol-induced contraction in guinea-pig urinary bladder strips and significant binding to muscarinic receptors.
- Acts as a muscarinic acetylcholine receptor (mAChR) antagonist
- Active metabolite of Tolterodine
- Inhibits carbachol-induced contraction of isolated guinea-pig urinary bladder strips
- Exhibits significant binding activity to muscarinic receptors in various tissues, with a longer duration in the bladder
- Suitable for overactive bladder research
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