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Medchemexpress LLC (Rac)-Acolbifene (EM-343; (Rac)-EM-652) | 151533-34-5 | 98.2% | 457.56 | 1 ML
Supplier: Medchemexpress LLC HY16023B10MM/1ML
(Rac)-Acolbifene (EM-343; (Rac)-EM-652) is the racemic form of EM652, an estrogen receptor antagonist, exhibiting both anti-estrogenic and estrogenic activities. This compound contains a piperidine ring and demonstrates a good pharmacological profile with a relative binding affinity (RBA) of 380. It shows an inhibitory effect in T-47D cells and antiuterotrophic inhibitions in ovariectomized mice.
- Racemic form of EM652.
- Acts as an estrogen receptor antagonist.
- Exhibits anti-estrogenic and estrogenic activities.
- Contains a piperidine ring.
- Demonstrates a good pharmacological profile with a relative binding affinity (RBA) of 380.
- Inhibits T-47D cell growth with an IC50 value of 0.110 nM.
- Induces antiuterotrophic inhibitions in ovariectomized mice.
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